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Publication date Communities Collections Article title Author(s) Journal/Conference
26 Mar 2026 Others Experimental Drug Development Centre In Silico‐Enabled Discovery and Development of Potent and Selective CDK11 Inhibitors (Pending publish) Frankie S. Mak, Fui Mee Ng, Padmanabhan Anbazhagan, Vikas Madan, Qian Wen Tan, Yiyang See, Diane Lim, Frances Karla Kusuma, Hannah Toh, Juliana Mohammad, Haiyan Yang, Sandra Sim, Li Hong Tan, Eileen Tay, Ronald Toh Kuan Hai, Perlyn Zekui Kwek, Mei Yee Wong, Deepika Raman, Qi An Ang, Vithya Manoharan, Susmitha Vuddagiri, Monique Danielle Dawson, Alison Tan, Joma Kanikadu Joy, Bong Hwa Gan, Choon Bing Low, Haoying Xu, Siew Pheng Lim, Hannes Hentze, Joseph Cherian, Chong Teik Tan, Jackie Ang, Kantharaj Ethirajulu, Klement Foo, Inderjeet Singh, Weijun Xu ChemMedChem
7 Aug 2025 Others Experimental Drug Development Centre Discovery of an Orally Bioavailable Reversible Covalent SARS-CoV-2 Mpro Inhibitor with Pan-Coronavirus Activity Qian Wen Tan, Subramanyam Vankadara, Jia Yi Fong, Yi Yang See, Nithya Baburajendran, Pearly Shuyi Ng, Weijun Xu, Yee Khoon Yeo, Weiling Wang, Choon Heng Low, Li Hong Tan, Eileen Gui Ju Tay, Yun Xuan Wong, Chuhui Huang, Sandra Sim, Shi Hua Ang, Hannah Hui Min Toh, Juliana Mohammad, Gang Wang, Boping Liu, Shu Ting Tan, Perlyn Zekui Kwek, Monique Danielle Dawson, Qin Yao Oh, Xiaoying Koh, Joma Joy, May Ann Lee, Walter Stunkel, Vishal Pendharkar, Hannes Hentze, Siew Pheng Lim, Kantharaj Ethirajulu, C. S. Brian Chia, Joseph Cherian Journal of Medicinal Chemistry
30 Oct 2024 Others Experimental Drug Development Centre Button-Push On-Demand Synthesis for Rapid Optimization of Antiviral Peptidomimetics Duanshuai Tian, Ting Wei Tan, Ronald Toh Kuan Hai, Gan Wang, Fadhil Peer Mohamed, Zhenyang Yu, Hwee Ting Ang, Weijun Xu, Qian Wen Tan, Pearly Shuyi Ng, Choon Heng Low, Boping Liu, Perlyn Quek Zekui, Joma Kanikadu Joy, Joseph Cherian, Frankie S Mak, Jie Wu Journal of the American Chemical Society
15 Feb 2024 Others Experimental Drug Development Centre Identification of small‐molecule binding sites of a ubiquitin‐conjugating enzyme‐UBE2T through fragment‐based screening Yong Yao Loh, Jothi Anantharajan, Qiwei Huang, Weijun Xu, Justina Fulwood, Hui Qi Ng, Elizabeth Yihui Ng, Chong Yu Gea, Meng Ling Choong, Qian Wen Tan, Xiaoying Koh, Wan Hsin Lim, Kassoum Nacro, Joseph Cherian, Nithya Baburajendran, Zhiyuan Ke, CongBao Kang Protein Science
11 Nov 2023 Others Experimental Drug Development Centre Identification and characterization of inhibitors covalently modifying catalytic cysteine of UBE2T and blocking ubiquitin transfer Jothi Anantharajan, Qian Wen Tan, Justina Fulwood, Wang Sifang, Qiwei Huang, Hui Qi Ng, Xiaoying Koh, Weijun Xu, Joseph Cherian, Nithya Baburajendran, CongBao Kang, Zhiyuan Ke Biochemical and Biophysical Research Communications
19 Jul 2022 Others Experimental Drug Development Centre A Warhead Substitution Study on the Coronavirus Main Protease Inhibitor Nirmatrelvir Subramanyam Vankadara, Monique Danielle Dawson, Jia Yi Fong, Qin Yao Oh, Qi An Ang, Boping Liu, Hong Yun Chang, Judice Koh, Xiaoying Koh, Qian Wen Tan, Joma Joy, Cheng San Brian Chia ACS Medicinal Chemistry Letters
14 Jul 2021 Others Experimental Drug Development Centre A head-to-head comparison of the inhibitory activities of 15 peptidomimetic SARS-CoV-2 3CLpro inhibitors Subramanyam Vankadara, Yun Xuan Wong, Boping Liu, Yi Yang See, Li Hong Tan, Qian Wen Tan, Gang Wang, Ratna Karuna, Xue Guo, Shu Ting Tan, Jia Yi Fong, Joma Joy, C.S. Brian Chia Bioorganic & Medicinal Chemistry Letters