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15 Feb 2024 Others Experimental Drug Development Centre Identification of small‐molecule binding sites of a ubiquitin‐conjugating enzyme‐UBE2T through fragment‐based screening Yong Yao Loh, Jothi Anantharajan, Qiwei Huang, Weijun Xu, Justina Fulwood, Hui Qi Ng, Elizabeth Yihui Ng, Chong Yu Gea, Meng Ling Choong, Qian Wen Tan, Xiaoying Koh, Wan Hsin Lim, Kassoum Nacro, Joseph Cherian, Nithya Baburajendran, Zhiyuan Ke, CongBao Kang Protein Science
11 Nov 2023 Others Experimental Drug Development Centre Identification and characterization of inhibitors covalently modifying catalytic cysteine of UBE2T and blocking ubiquitin transfer Jothi Anantharajan, Qian Wen Tan, Justina Fulwood, Wang Sifang, Qiwei Huang, Hui Qi Ng, Xiaoying Koh, Weijun Xu, Joseph Cherian, Nithya Baburajendran, CongBao Kang, Zhiyuan Ke Biochemical and Biophysical Research Communications
19 Jul 2022 Others Experimental Drug Development Centre A Warhead Substitution Study on the Coronavirus Main Protease Inhibitor Nirmatrelvir Subramanyam Vankadara, Monique Danielle Dawson, Jia Yi Fong, Qin Yao Oh, Qi An Ang, Boping Liu, Hong Yun Chang, Judice Koh, Xiaoying Koh, Qian Wen Tan, Joma Joy, Cheng San Brian Chia ACS Medicinal Chemistry Letters
14 Jul 2021 Others Experimental Drug Development Centre A head-to-head comparison of the inhibitory activities of 15 peptidomimetic SARS-CoV-2 3CLpro inhibitors Subramanyam Vankadara, Yun Xuan Wong, Boping Liu, Yi Yang See, Li Hong Tan, Qian Wen Tan, Gang Wang, Ratna Karuna, Xue Guo, Shu Ting Tan, Jia Yi Fong, Joma Joy, C.S. Brian Chia Bioorganic & Medicinal Chemistry Letters