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14 Nov 2020 BMRC Singapore Institute of Food and Biotechnology Innovation In-Silico Identified New Natural Sortase A Inhibitors Disrupt S. aureus Biofilm Formation Chung Yan Leong, Veronica Ng, Yoganathan Kanagasundaram, Hao Fan, Siew Bee Ng, Kishore Reddy Venkata Thappeta, Li Na Zhao, Choy Eng Nge, Sharon Crasta International Journal of Molecular Sciences
28 Feb 2020 BMRC Bioinformatics Institute Viruses go modular Ariel Shepley-McTaggart, Hao Fan, Marius Sudol, Ronald N. Harty Journal of Biological Chemistry
6 Sep 2019 BMRC Bioinformatics Institute Reviewing HIV-1 Gag Mutations in Protease Inhibitors Resistance: Insights for Possible Novel Gag Inhibitor Designs Chinh Tran-To Su, Darius Wen-Shuo Koh, Samuel Ken-En Gan Molecules
30 May 2019 BMRC p53 Laboratory Stereoisomerism of Stapled Peptide Inhibitors of the p53-Mdm2 Interaction: An Assessment of Synthetic Strategies and Activity Profiles Tsz Ying Yuen, Christopher J. Brown, Yuezhen Xue, Yaw Sing Tan, Fernando J. Ferrer Gago, Xue Er Lee, Jin Yong Neo, Dawn Thean, Hung Yi Kristal Kaan, Anthony W. Partridge, Chandra S. Verma, David P. Lane, Charles W. Johannes Chemical Science
28 May 2019 BMRC Bioinformatics Institute Preclinical Characteristics of the Irreversible Pan-HER Kinase Inhibitor Neratinib Compared with Lapatinib: Implications for the Treatment of HER2-Positive and HER2-Mutated Breast Cancer Denis M. Collins, Neil T. Conlon, Srinivasaraghavan Kannan, Chandra S. Verma, Lisa D. Eli, Alshad S. Lalani, John Crown Cancers
30 Aug 2018 BMRC p53 Laboratory Synthetic 10FN3-based mono- and bivalent inhibitors of MDM2/X function S. Y. Lau, J. W. Siau, R. M. Sobota, C. I. Wang, P. Zhong, D. P. Lane, F. J. Ghadessy Protein Engineering, Design & Selection
12 Jul 2018 BMRC Bioinformatics Institute Homologous Lympho-Epithelial Kazal-type Inhibitor Domains Delay Blood Coagulation by Inhibiting Factor X and XI with Differential Specificity Karthik Ramesh, Dilraj Lama, Kang Wei Tan, Van Sang Nguyen, Fook Tim Chew, Chandra S. Verma, Yu Keung Mok Structure
3 Jul 2018 BMRC Bioinformatics Institute Global update on the susceptibility of human influenza viruses to neuraminidase inhibitors and status of novel antivirals, 2016-2017. Angie Lackenby, Terry G. Besselaar, Rod S. Daniels, Alicia Fry, Vicki Gregory, Larisa V. Gubareva, Weijuan Huang, Aeron C. Hurt, Sook-Kwan Leang, Raphael T. C. Lee, Janice Lo, Lori Lollis, Sebastian Maurer-Stroh, Takato Odagiri, Dmitriy Pereyaslov, Emi Takashita, Dayan Wang, Wenqing Zhang, Adam Meijer Antiviral Research
16 Mar 2018 BMRC p53 Laboratory A DHODH Inhibitor Increases p53 Synthesis and Enhances Tumor Cell Killing by p53 Degradation Blockage Marcus J. G. W. Ladds, Ingeborg M. M. van Leeuwen, Catherine J. Drummond, Su Chu, Alan R. Healy, Gergana Popova, Andrés Pastor Fernández, Tanzina Mollick, Mihaela Popa, Suhas Darekar, Saikiran K. Sedimbi, Marta Nekulova, Marijke C. C. Sachweh, Johanna Campbell, Maureen Higgins, Chloe Tuck, Mireia Mayoral Safont, Pascal Gelebart, Zinayida Fandalyuk, Alastair M. Thompson, Richard Svensson, Anna-Lena Gustavsson, Lars Johansson, Katarina Färnegårdh, Ulrika Yngve, Aljona Saleh, Martin Haraldsson, Agathe C. A. D'Hollander, Marcela Franco, Yan Zhao, Maria Håkansson, Björn Walse, Karin Larsson, Emma M. Peat, Vicent Pelechano, John Lunec, Borivoj Vojtesek, Mar Carmena, William C. Earnshaw, Anna R. McCarthy, Nicholas J. Westwood, Marie Arsenian-Henriksson, David P. Lane, Ravi Bhatia, Emmet McCormack, Sonia Lain Nature Communications
9 Nov 2017 BMRC p53 Laboratory A yeast two-hybrid system for the screening and characterization of small-molecule inhibitors of protein–protein interactions identifies a novel putative Mdm2-binding site in p53 Jin Huei Wong, Mohammad Alfatah, Mei Fang Sin, Hong May Sim, Chandra S. Verma, David P. Lane, Prakash Arumugam BMC Biology