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7 Aug 2025
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Experimental Drug Development Centre
Discovery of an Orally Bioavailable Reversible Covalent SARS-CoV-2 Mpro Inhibitor with Pan-Coronavirus Activity
Qian Wen Tan,
Subramanyam Vankadara,
Jia Yi Fong,
Yi Yang See,
Nithya Baburajendran,
Pearly Shuyi Ng,
Weijun Xu,
Yee Khoon Yeo,
Weiling Wang,
Choon Heng Low,
Li Hong Tan,
Eileen Gui Ju Tay,
Yun Xuan Wong,
Chuhui Huang,
Sandra Sim,
Shi Hua Ang,
Hannah Hui Min Toh,
Juliana Mohammad,
Gang Wang,
Boping Liu,
Shu Ting Tan,
Perlyn Zekui Kwek,
Monique Danielle Dawson,
Qin Yao Oh,
Xiaoying Koh,
Joma Joy,
May Ann Lee,
Walter Stunkel,
Vishal Pendharkar,
Hannes Hentze,
Siew Pheng Lim,
Kantharaj Ethirajulu,
C. S. Brian Chia,
Joseph Cherian
Journal of Medicinal Chemistry
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