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7 Aug 2025
Others
Experimental Drug Development Centre
Discovery of an Orally Bioavailable Reversible Covalent SARS-CoV-2 Mpro Inhibitor with Pan-Coronavirus Activity
Qian Wen Tan,
Subramanyam Vankadara,
Jia Yi Fong,
Yi Yang See,
Nithya Baburajendran,
Pearly Shuyi Ng,
Weijun Xu,
Yee Khoon Yeo,
Weiling Wang,
Choon Heng Low,
Li Hong Tan,
Eileen Gui Ju Tay,
Yun Xuan Wong,
Chuhui Huang,
Sandra Sim,
Shi Hua Ang,
Hannah Hui Min Toh,
Juliana Mohammad,
Gang Wang,
Boping Liu,
Shu Ting Tan,
Perlyn Zekui Kwek,
Monique Danielle Dawson,
Qin Yao Oh,
Xiaoying Koh,
Joma Joy,
May Ann Lee,
Walter Stunkel,
Vishal Pendharkar,
Hannes Hentze,
Siew Pheng Lim,
Kantharaj Ethirajulu,
C. S. Brian Chia,
Joseph Cherian
Journal of Medicinal Chemistry
25 Apr 2025
Others
Experimental Drug Development Centre
Structure-based discovery of novel non-covalent small molecule inhibitors of USP30
Padmanabhan Anbazhagan,
Jothi Anantharajan,
Justina Fulwood,
Choon Heng Low,
Nithya Baburajendran,
Klement Foo,
Weijun Xu
Journal of Computer-Aided Molecular Design
30 Oct 2024
Others
Experimental Drug Development Centre
Button-Push On-Demand Synthesis for Rapid Optimization of Antiviral Peptidomimetics
Duanshuai Tian,
Ting Wei Tan,
Ronald Toh Kuan Hai,
Gan Wang,
Fadhil Peer Mohamed,
Zhenyang Yu,
Hwee Ting Ang,
Weijun Xu,
Qian Wen Tan,
Pearly Shuyi Ng,
Choon Heng Low,
Boping Liu,
Perlyn Quek Zekui,
Joma Kanikadu Joy,
Joseph Cherian,
Frankie S Mak,
Jie Wu
Journal of the American Chemical Society
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