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7 Jun 2019
Others
Experimental Drug Development Centre
Backbone resonance assignment for the full length tRNA-(N1G37) methyltransferase of Pseudomonas aeruginosa
Yan Li,
Wenhe Zhong,
Ann Zhufang Koay,
Hui Qi Ng,
Qianhui Nah,
Yee Hwa Wong,
Jeffrey Hill,
Julien Lescar,
Peter C. Dedon,
CongBao Kang
Biomolecular NMR Assignments
23 May 2019
Others
Experimental Drug Development Centre
Discovery of Irreversible Inhibitors Targeting Histone Methyltrans-ferase, SMYD3
Chuhui Huang,
Si Si Liew,
Grace R Lin,
Anders Poulsen,
Melgious J. Y. Ang,
Brian C. S. Chia,
Sin Yin Chew,
Zekui Perlyn Kwek,
John L. K. Wee,
Esther H. Ong,
Priya Retna,
Nithya Baburajendran,
Rong Li,
Weixuan Yu,
Xiaoying Koh-Stenta,
Anna Ngo,
Sravanthy Manesh,
Justina Fulwood,
Zhiyuan Ke,
Hwa Hwa Chung,
Sugunavathi Sepramaniam,
Xin Hui Chew,
Nurul Dinie,
Yun Shan Chew,
May Ann Lee,
Choon Bing Low,
Vishal Pendharkar,
Vithya Manoharan,
Susmitha Vuddagiri,
Kanda Sangthongpitag,
Joma Joy,
Alex Matter,
Jeffrey Hill,
Thomas Keller,
Klement Foo
ACS Medicinal Chemistry Letters
8 Oct 2018
Others
Experimental Drug Development Centre
Backbone resonance assignment for the N-terminal region of bacterial tRNA-(N1G37) methyltransferase
Yan Li,
Wenhe Zhong,
Ann Zhufang Koay,
Hui Qi Ng,
Xiaoying Koh-Stenta,
Qianhui Nah,
Siau Hoi Lim,
Andreas Larsson,
Julien Lescar,
Jeffrey Hill,
Peter C. Dedon,
CongBao Kang
Biomolecular NMR Assignments
13 Aug 2018
Others
Experimental Drug Development Centre
Designing an ultra-short antibacterial peptide with potent activity against Mupirocin-resistant MRSA
Giovinna Arfan,
Chu Yang Fann Ong,
Siew Mei Samantha Ng,
Qiu Ying Lau,
Fui Mee Ng,
Esther Hong Qian Ong,
Jeffrey Hill,
Cheng San Brian Chia
Chemical Biology & Drug Design
11 Aug 2018
Others
Experimental Drug Development Centre
Discovery of dual GyrB/ParE inhibitors active against Gram-negative bacteria
Soo Yei Ho,
Weiling Wang,
Fui Mee Ng,
Yun Xuan Wong,
Zhi Ying Poh,
Wai Sum Eldwin Tan,
Shi Hua Ang,
Si Si Liew,
Yin Sze Joyner Wong,
Yvonne Tan,
Anders Poulsen,
Vishal Pendharkar,
Kanda Sangthongpitag,
John Manchester,
Gregory Basarab,
Jeffrey Hill,
Thomas H. Keller,
Joseph Cherian
European Journal of Medicinal Chemistry
5 Jul 2018
BMRC
Bioinformatics Institute
Targeting cancer addiction for SALL4 by shifting its transcriptome with a pharmacologic peptide
Bee Hui Liu,
Chacko Jobichen,
C. S. Brian Chia,
Tim Hon Man Chan,
Jing Ping Tang,
Theodora X. Y. Chung,
Jia Li,
Anders Poulsen,
Alvin W. Hung,
Xiaoying Koh-Stenta,
Yaw Sing Tan,
Chandra S. Verma,
Hong Kee Tan,
Chan-shuo Wu,
Feng Li,
Jeffrey Hill,
Joma Joy,
Henry Yang,
Li Chai,
J. Sivaraman,
Daniel G. Tenen
Proceedings of the National Academy of Sciences
5 Jul 2018
Others
Experimental Drug Development Centre
Targeting cancer addiction for SALL4 by shifting its transcriptome with a pharmacologic peptide
Bee Hui Liu,
Chacko Jobichen,
Cheng San Brian Chia,
Tim Hon Man Chan,
Jing Ping Tang,
Theodora Chung,
Jia Li,
Anders Poulsen,
Alvin W. Hung,
Xiaoying Koh-Stenta,
Yaw Sing Tan,
Chandra S. Verma,
Hong Kee Tan,
Chan-shuo Wu,
Feng Li,
Jeffrey Hill,
Joma Joy,
Henry Yang,
Li Chai,
J. Sivaraman,
Daniel G. Tenen
PNAS
23 May 2018
Others
Experimental Drug Development Centre
Structural and ligand binding analysis of the YAP-binding domain of transcription factor TEAD4
Yan Li,
Shuang Liu,
Elizabeth Yihui Ng,
Rong Li,
Anders Poulsen,
Jeffrey Hill,
CongBao Kang,
Ajaybabu Pobbati,
Alvin Wei Hung,
Wanjin Hong,
Thomas Keller
Biochemical Journal
24 Apr 2018
Others
Experimental Drug Development Centre
Fragment-based drug discovery of potent Protein Kinase C-iota inhibitors
Jacek Kwiatkowski,
Boping Liu,
Doris Hui Ying Tee,
Guoying Chen,
Nur Huda Binte Ahmad,
Yun Xuan Wong,
Zhi Ying Poh,
Shi Hua Ang,
Eldwin Sum Wai Tan,
Esther Ong,
Nurul Dinie,
Anders Poulsen,
Vishal Pendharkar,
Kanda Sangthongpitag,
May Ann Lee,
Sugunavathi D/O Sepramaniam,
Soo Yei Ho,
Joseph Cherian,
Jeffrey Hill,
Thomas Hugo Keller,
Alvin Wei Hung
Journal of Medicinal Chemistry
23 Apr 2018
BMRC
Bioinformatics Institute
Optimization of Selective Mitogen-Activated Protein Kinase Interacting Kinases 1 and 2 Inhibitors for the Treatment of Blast Crisis Leukemia
Haiyan Yang,
Lohitha Rao Chennamaneni,
Melvyn Wai Tuck Ho,
Shi Hua Ang,
Eldwin Sum Wai Tan,
Duraiswamy Athisayamani Jeyaraj,
Yoon Sheng Yeap,
Boping Liu,
Esther Hq Ong,
Joma Kanikadu Joy,
John Liang Kuan Wee,
Perlyn Kwek,
Priya Retna,
Nurul Dinie,
Thuy Thi Hanh Nguyen,
Shi Jing Tai,
Vithya Manoharan,
Vishal Pendharkar,
Choon Bing Low,
Yun Shan Chew,
Susmitha Vuddagiri,
Kanda Sangthongpitag,
Meng Ling Choong,
May Ann Lee,
Srinivasaraghavan Kannan,
Chandra S. Verma,
Anders Poulsen,
Sharon Lim,
Charles Chuah,
Tiong Sin Ong,
Jeffrey Hill,
Alex Matter,
Kassoum Nacro
Journal of Medicinal Chemistry
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